NEW! Silverback Labs GW501516 Oral Dropper Solution with pipette 25mg/ml - 30ml bottle

£35.00

  • Product Code: sbgw5
  • Availability: In Stock
  • Ex Tax: £35.00

Tags: NEW! Silverback Labs GW501516 Oral Dropper Solution with pipette 25mg/ml - 30ml bottle

NEW & EXCLUSIVE! Made and sold in the United Kingdom, we are now for the exclusive distributors for Silverback Labs.


GW-501516 (GW1516, Endurobol or GSK-516) acts as a PPAR-β modulator. GW 501516 activates AMP-activated protein kinase and stimulates glucose uptake in skeletal muscle tissue, and GW-501516 has been demonstrated to reverse metabolic abnormalities in obese mice with pre-diabetic metabolic syndrome, most likely by stimulating fatty acid oxidation.

           PPAR-β modulator

           Agitate bottle before each administration

           Not for human consumption

 

GW50156 regulates fat burning through a number of mechanisms. It increases glucose uptake in skeletal muscle tissue and increases muscle gene expression, especially genes involved in preferential lipid utilization. This shift changes the body's metabolism to favour burning fat for energy instead of carbohydrates or muscle protein, potentially allowing clinical application for obese patients to lose fat effectively without experiencing muscle catabolism or the effects and satiety issues associated with low blood sugar. GW-501516 also increases muscle mass, which improved glucose tolerance and reduced fat mass accumulation even in mice fed a very high fat diet, suggesting that GW-501516 may have a protective effect against obesity.

It has been demonstrated at an oral doses of just 5 mg a day to reverse metabolic abnormalities in obese mice with pre-diabetic metabolic syndrome, most likely by stimulating fatty acid oxidation. Treatments with GW-501516 have been also shown to increase HDL cholesterol by up to 79% in rhesus monkeys and the compound is now undergoing Phase II trials to improve HDL cholesterol.

M.Wt: 453.498

Formula: C21H18F3NO3S2 

Solubility: DMSO/CMC

Purity: >99%

Storage: at 20? 2 years

Half life: 24 hours

CAS No.: 317318-70-0

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